Utano, Gadziriro
Description uye mirayiridzo kushandiswa: "Albarel"
Chii chinodhaka "Albarel"? Mirayiridzo dzokushandisa uye tsanangudzo mushonga uyu ichakurukurwa pazasi. Nesuwo kukuudza pamusoro fomu umo zvinodhaka asunungurwa pane zviri kunoshamisa sei varwere vanoteerera.
Zvinoumba, tsananguro, chimiro
In Wakadiniko kugadzirwa pasi mishonga ongororo? Zvarinotaura pamusoro mirayiridzo kushandiswa? "Albarel" - rakatenderera, biconvex mahwendefa chena ruvara, iro vane achiita zvokutemera kumativi ose ari muchimiro «H» chiratidzo.
The mushonga rakazara muna Maronda akasiyana zvezvimedu 10 uye makadhibhokisi bhokisi, ukuwo.
Chii chinokonzera "Albarel" chinodhaka? Mirayiridzo yokushandisa inoshuma kuti mamiriro vanzwe kuti chokushandisa rilmenidine. Kunosanganisirawo vakaneta chishongedzo zvokubikisa sezvo yavaibvisa carboxymethyl starch, MCC, rakasimba Paraffin, lactose, magnesium stearate, colloidal anhydrous silica, talc uye wakisi chena.
pharmacology
Chii kunotaurwa mushonga? Zvarinotaura pamusoro mirayiridzo kushandiswa? "Albarel" ane antihypertensive mumiririri uye oxazoline rinobva.
Mushure kushandisa mishonga anopinda noukama imidazoline receptors ari peripheral uye cortical vasomotor nzvimbo, kusanganisira renal nzvimbo. rilmenidine kusakarongeka pamwe zvinhu izvi zvinobatsira kuti chinovhiringidza pamusoro peripheral sympathomimetic basa uye cortical nzvimbo, iyo pakupedzisira inotungamirira richikwidibira ropa nevezera.
Features zvinodhaka
Kugadzirira "Albarel" analogs, mirayiridzo kushandiswa zviri kukurukurwa hereinafter, ine hypotensive nomugumisiro (zvichienderana kugamuchirwa zvokurarama dosing) kuti systolic uye diastolic BP richimire kana nhema chinzvimbo. Zvinonzi kwakaratidza kuti vatarisire kuti mushonga pa kuchirapa mishonga (i.e., 1 kana 2 MG pazuva) dzinobudirira mukurapa mwero kune munyoro neBP.
Maererano nenyanzvi, nezvaizoitwa mumiririri uyu kunochengetwa masikati. Uyezve, zviri abudirire panguva yechiitwa.
Refu kushandiswa kwezvinodhaka haakonzeri muropa.
ehupfumi zvinodhaka
Chii chinoshamisa ndiyo nzira se "Albarel"? Mirayiridzo yokushandisa, nyanzvi chaidzo vanotaura kuti zvinodhaka izvi panguva kuchirapa mishonga haadi kuchinja kushanda mwoyo, uye asingadi kuti kunonoka remvura yavaibvisa mumuviri uye asingauyi kunokanganisa metabolic nomwero.
mushonga uyu kunoderedza peripheral vascular nemishonga pasina shanduko ipi cardiac goho. Zvinofanira kucherechedzwa kuti electrophysiological maindex uye myocardial contractility pavarwere kugamuchira zvinodhaka ichi kuramba kuchinja.
Vaiona antihypertensive mushonga haakonzeri orthostatic hypotension (kusanganisira vakwegura), haana kumbochinja ropa aibuda renal, usingasii kunokanganisa vasiri siyana (compensatory) mwoyo zvazvingava pamusoro muviri, uye hazvina chokuita mafuta uye carbohydrate Exchange, filtration chakapatsanurwa uye glomerular filtration.
kinetics
Ko "Albarel" mapiritsi vari kunyura? Mirayiridzo Dzokushandisa rinoti kuti mushonga akati iri zvachose uye nokukurumidza woga kubva ura. Pashure chete dose aona pashure 2 chasa ayo kunonyanyisa zvinodhaka wevasungwa munguva plasma.
The Mhedziso bioavailability zvinodhaka riri 100%. Zvinofanira kucherechedzwa kuti hazvina pasi kutanga nomunyika chiropa.
The zvakanyatsoenzana mamiriro murwere yakasimbiswa chete pazuva dzose yaunodya mahwendefa rechitatu. Vanhu vane BP vari kurapwa kwemakore, wevasungwa zvinodhaka munyika yeplasma akatsiga.
mushonga Izvi yabudiswa muna mukaka. metabolites Its inowanikwa weti chete chero mari. hafu-upenyu zvinodhaka zvinotora maawa anenge 8. Nguva iyi haachinji kunyange kana apiwa kugadzwa pamahwendefa.
umboo
Mune zvimwe zviitiko, mushonga wacho ushandiswe varwere vaiona? Zvarinotaura pamusoro mirayiridzo kushandiswa? "Albarel" - chiri antihypertensive mumiririri, iro achishingaira kushandiswa neBP.
Kurambidzwa kugadzwa
Kushandiswa kwezvinodhaka "Albarel" hakubvumidzwi mu:
- pamuviri;
- nokuora mwoyo;
- renal kukundikana (kwazvo);
- achiyamwa;
- Hypersensitivity kuti rilmenidine kana zvimwe zvinoumba chezvinodhaka.
Zvinofanira kucherechedzwa kuti mishonga iyi haina kushandiswa chiremba tsika.
Mahwendefa "Albarel": mirayiridzo kushandiswa
Mabatirwo chokushandisa ichi zvinofanira chokugutsikana chete pashure zano chiremba. Kana murwere zvisingaiti kubvunza chiremba wako usati kutora mushonga vanofanira kuverenga nokungwarira mirayiridzo. Maererano naye, kuitira kuti vabudirire zvinozoita, murwere zvakakwana kutora rimwe piritsi asati adya. Kana chipimo chemushonga ichi "Albarel" haana kuvandudza mamiriro murwere, ipapo yakawedzera kusvika 2 Mahwendefa pazuva (kutora zuva asati zvemangwanani uye chisvusvuro).
vaiona nzira yokurapa-refu.
Pasinei nokuti abolition mishonga iyi hakuiti kazhinji kukonzera marwadzo, discontinuation yokurapa kunofanira kuva zvishoma nezvishoma, pamwe zvishoma nezvishoma zvinoderedza dose.
Zviito ne-hunhu
Ndezvipi kumativi Migumisiro anonzi antihypertensive mumiririri? Zvakadini anoti mirayiridzo kushandiswa? "Albarel" kungakonzera zvakadai zvisingadiwi mananara se:
- palpitations, orthostatic hypotension, migumisiro chando wamativi (mu zvisingawanzoitiki zviitiko);
- asthenia, vakawedzera kuneta panguva yechiitwa, hope, kufunganya, kushaya hope kana kuora mwoyo, nokugwinha (mu zvisingawanzoitiki zviitiko);
- kuda kurutsa, epigastric marwadzo, kupatira, kuoma iri mumuromo, manyoka;
- kuvaviwa, ganda nekumhanyirira.
Tinofanirawo kuziva kuti apo kunwa mushonga uyu, vamwe varwere ruzivo peripheral edema, kupiswa uye zvepabonde dysfunction.
ovhadhozi rinoreva
Chii chichaitika kana uchishandisa vazhinji "Albarel" Mahwendefa? Mirayiridzo yokushandisa, mishonga kuti mumiririri uyu kunge kukurukurwa pamusoro. Kana iwe kusapfuudza wokupedzisira murwere anogona kuva chakakomba hypotension uye kutyorwa-siyana mune psyche. Panyaya iyi, munhu basa gastric lavage uye akatakura sympathomimetic kurapa.
Kudyidzana nevamwe zvinodhaka
Hazvina varumbidzwa kutora "Albarel" mapiritsi pamwe doro uye Mao FIs. zvinotevera zvinoratidza vaiona zvinodhaka zvinodhaka mukukurukurirana vave kuzivikanwa senyanzvi:
- pamwe diuretics, antihistamines uye vasodilators kunoitika potentiation mugumisiro zvinodhaka;
- pamwe tricyclic antidepressants akacherekedza kuderera antihypertensive mugumisiro zvinodhaka;
- zvinodhaka kuti tunodzivisa zviito nechepakati tsinga, vakawedzera Kurara kuchengetwa.
chaicho mashoko
Kana mushonga rinoshandiswa vanhu vachangobva nesitiroko kana myocardial infarction, kwavari Zvinoda kuramba kurapwa achitarisirwa.
Tichifunga akanaka kubvumirawo zvimwe mahwendefa 'Albarel "rinogona kushandiswa varwere vakwegura uye varwere chirwere cheshuga mellitus.
Kana uchida kumisa kurapwa, zvinodhaka chipimo chemushonga anofanira kuderedzwa zvishoma nezvishoma. Zvinofanira kurangarirwa kuti kakawanda, ari abolition zvinodhaka hakuna pamwe chero nemishonga.
It hakubvumidzwi kuti ndipe "Albarel" panguva imwe chete Mao FIs uye doro tubhokisi zvigadzirwa.
Clinical mashoko pamusoro efficacy uye kuchengeteka mishonga muvana uye vechiduku hakuna kukwana. Panyaya iyi, akarayira kuti mushonga varwere izvi hazvifaniri kuva.
At kuchirapa mishonga "Albarel" haana kumbochinja psychomotor siyana kwevanhu. Kana mushonga zvakapfuudzwa vazhinji kana zvinodhaka, kudzvinyirira nechepakati tsinga basa, umo nyaya murwere hakubvumidzwi kutyaira motokari, uyewo kuita mamwe mabasa ngozi.
Analogs uye nhoroondo
Analogs atakurukura zvinodhaka hakusi kwazvo. Zvezvisarudzo kutengeka uye inonyanya kufarirwa vari "Tenaksum". medicament Ichi antihypertensive mumiririri kuva boka oxazolines. Ane zvakafanana mazita contraindications uye marwadzo, asi zvakawanda zvinodhura.
With Panyaya zvakataurwa varwere pamusoro zvinodhaka ichi, vari vashoma. Kufanana vanachiremba, vatengi vanoti kuti inoshanda chaizvo nzira kubvisa neBP. Kana zvemashoko zvinodhaka zvinosanganisira kwayo kwenguva refu kuchirapa zvazviri, kusanganisira panguva yechiitwa.
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