Utano, Gadziriro
Mapiritsi ari kufurirwa "Fiziotenz": mhinduro wevarwere uye vanachiremba
Inoshanda antihypertensive mushonga, munhu anosarudza imidazoline Kanotokonya agonist chinhu chinodhaka "Fiziotenz". Testimonials vanoti zvinoreva zvinobatsira kudzibatsira kuti chirwere cheshuga uye vanhu rurefu body mass.
neBP Features
Zvirwere zvomwoyo uye ropa midziyo inozviisa vazhinji. Zvisinei, mune vakadzi zvarakasiya izvi pave paya kupfuura vanhu. Asi ivo kuitika zvikuru kwakatooma uye inozivikanwa dzakakwirira dziine BP, kunyanya raidudzwa dzinorwadza zviratidzo. NeBP kazhinji anovandudza nevamwe pathologies: kufutisa, chirwere cheshuga, zvirwere chiropa uye itsvo kukundikana lipid muviri.
Pamwe chete kuwedzera body mass kunoitika nokuvhiringidzirwa SNA, unova kukonzera cheBP uye BP inotungamirwa. Dzinounzwa symptomatic tsinga mahormone mipiro luminal aienda rwengarava ropa, zvichiguma mwoyo pakukurukura reokisijeni kuti nyama uye nhengo vane kusunda ropa kuti torque pasi kumusoro kumanikidzwa, saka kuva BP, izvo chinoita vaitire mishonga nzira. Mumwe zvinodhaka, vachibvumira yakawedzera kuomesa mumugwagwa, inzira "Fiziotenz".
Mamiriro uye Kuronga
Yakabudiswa medicament muchimiro mahwendefa film-zvemapuranga. Huru achishingaira fuma mabasa moksonindin. Ebetsero zvinoriumba zvinosanganisira magnesium stearate, crospovidone, povidone, lactose monohydrate.
pharmacological ehupfumi
The kushingaira zvacho medicament ane musimboti hypotensive chiito. Moxonidine muuropi hunde masero zvokusarudza kunomutsa kutsinga dzinouya receptors, izvo zvinobatanidzwa mutemo tonic dzepanguva uye symptomatic tsinga. Zvinoguma vasanyanye basa uye symptomatic peripheral arterial nevezera. zveBhaibheri zvakawanda (kurapa kunonyaradza pfungwa raitungamirirwa, randomized, kaviri-bofu) zvinoratidza kubudirira zvinodhaka "Fiziotenz". Reviews wevarwere vanosimbisa kuti mushonga kusiyana nemamwe sympatholytic antihypertensive yomuchipatara kuti murege kukonzera muromo yakaoma, kana rinoshandiswa hapana nyaradzo.
Pharmacodynamics uye Pharmacokinetics
Mushure yomukati kugamuchirwa zvinoreva 90 muzana woga kubva gastro-intestinal hurongwa. The kunonyanyisa wevasungwa yezviri fuma iri plasma iri kuchengetwa neawa. Meal pamusoro pharmacokinetics ose moxonidine une maturo.
Chikuru metabolite vanoshingaira remubatanidzwa iri dehydrogenated moxonidine uye guanidine nomukaka. Hafu-upenyu moxonidine kunoitika mumaawa 2,5 uye zuva nenguva 90% goho chinhu kuburikidza neitsvo ura.
In varwere BP, zvichienzaniswa nevanhu hwakanaka, kuchinja pharmacokinetics ose moxonidine vaizivikanwa. Zvishoma kinetic parameters zvinogona dzakachinjwa Varwere vakwegura inobatanidzwa zvinoderedza kunyatsoita muviri moksodinina, uyewo yaro bioavailability yepamusorosoro.
Drug "Fiziotenz" Mirayiridzo Use
Testimonials vanoti kuti mahwendefa anofanira kutorwa nemuromo zvisinei zvokudya zvinodyiwa. Kazhinji, mushonga inoshandiswa kwokutanga zuva chipimo chemushonga kuti 200 mcg. Kufadza kuroorwa Huwandu zvinodhaka haafaniri kupfuudza micrograms 400 zuva nezuva mari yakakamurwa nezvikwiriso zviviri - 600 micrograms. Varwere zvine mwero kuti zvikuru mwoyo kutadza vari pamusoro hemodialysis, Zvinokurudzirwa kutora micrograms 200 rimwe zuva rinoreva. Nezvakanaka kushivirira chitsama zvinodhaka anogona ngazviwedzerwe kaviri.
ovhadhozi
Kana kushandiswa kunyanyisa-siyana kunaka zvingaratidza kuitika zvinodhaka. Saka, mahwendefa kubva "Fiziotenz" kumanikidzwa (wongororo zvinoratidza izvozvo) kungamutsawo nomusoro, hope, nyaradzo. Kana chipimo chemushonga akapfuudza kufurirwa anogona rabada zvinokosha, kukudziridza marwadzo ari epigastric vakachengeta xerostomia, bradycardia, kurutsa, kurukutika, wakawedzera kurukutika, dzungu. Uyezve, varwere vanogona kuva nehanya hyperglycemia, tachycardia, uye zvinopfuura kuwedzera kumanikidza.
dzakananga mushonga yambokurukurwa nekuda pakurapa zviratidzo ovhadhozi. Kana hypotension anofanira kupinda dopamine uye kuwedzera mvura kugutsikana mumuviri. Zviratidzo bradycardia zvinokwanisika kurega kushandisa atropine. In ovhadhozi kuderedza kana kubvisa gangaidzo chirwere cheBP ashandise Arifa-adrenoceptor mhandu.
zvinodhaka kwavatori
Tikafunga zvinodhaka hapasi zvakafanira kukosha. Zvisinei, kana kugamuchira mbiri kana kupfuura zvinodhaka zvingava kwakaderera kana nokusimbaradza yakawiriranwa zviito. Muchiitiko chokutanga, mushonga hauchazopi akatarisirwa mugumisiro, mumamiriro ezvinhu wechipiri, pane mukana ane ovhadhozi, uye kunyange chepfu.
Saka, apo aishandisa zvinodhaka antihypertensive (thiazide diuretics, karusiyamu blockers anononoka Mipata) pamwe medicament "Fiziotenz" (wongororo kunyevera pamusoro ichi) zvingamuka hypotensive chirungiso maturo. Mawa kurapwa pamwe tricyclic antidepressant lowers kubudirira yapakati protivopertenzivnyh zvinodhaka, uye haafaniri kushandiswa pamwechete zvinodhaka "Fiziotenz".
Mukuwedzera, chishandiso unokubvumira kuvandudza zvishande basa pavarwere simba nokutanga zvinodhaka "Lorazepam". Application pamwe benzodiazepines kungaita kunowedzerwa nyaradzo. In kugadzwa zvinodhaka "Digoxin", "glibenclamide", "hydrochlorothiazide" hapana pharmacokinetic kudyidzana.
Shandisa panguva pamuviri
zvinodhaka Various kukanganisa fetus kana mudumbu, zvichitungamirira mune dzimwe nguva kune zvakaipa mwana. Sezvo zvinoumba zvinodhaka yatorwa mukaka waamai, anogona kuwira muviri mucheche uye kuita pairi. Naizvozvo, panguva yepamuviri uye lactation, zvakakodzera kutora zvakanyanyisa hanya mishonga.
Hakuna Kusara - uye zvinodhaka "Fiziotenz". Kugadzwa ake chinoshanda chete pashure zano nyanzvi, pokuongorora zvinogona kubatsira kuti amai uye kukuvadza mwana. Sezvo basa chirungiso zvinoenda mukaka panguva dzokudya mucheche vanofanira kusiya chikumbiro chacho kana kuti kurega uchiyamwisa.
zvidzidzo zvokuongorora kuitwa mhuka, zvakananga kana zvisina kunanga mugumisiro zvinodhaka riri pamuviri, fetus (embryo) kana postnatal kukura havana kuzivikanwa.
divi kushanda
Kufanana mishonga yakawanda, mapiritsi "Fiziotenz" (wongororo zvipupurire ichi) hunokonzera kusafarira kubva mumuviri. Izvi zvinowanzoitika kana ukashandisa kufadza mari kwenguva yakareba uye vari hypersensitive kuti zvinoshingaira chirungiso.
Tsinga ndiyo kushandiswa kwezvinodhaka ikasakendenga nemusoro, hope kana kushaya hope, dzungu. Zviratidzo izvi zvinoonekwa kakawanda. On chikamu mwoyo uye vascular gadziriro nenjodzi rwakavapo zvisingawanzoitiki kacho kunoratidzwa unopinza ichidonhedzera kumanikidzwa, orthostatic hypotension. Uyezve, varwere pashure muromo Kutarisirwa ruzivo yakaoma, kuda kurutsa, vanogona kuonekwa sechinhu dermatologic kuita angioedema, pruritus kana mapundu. Kana paine divi kushanda zvinodhaka harifaniri akamira, kunaka zviratidzo pashure pevhiki nhatu kushandiswa, avanotarisira kunyangarika. Zvisinei, bvunza nyanzvi ichiri kudikanwa.
Contraindications
Hapana mushonga "Fiziotenz" rinogona kutorwa nguva dzose. Reviews vanachiremba vanoti inokurudzirwa kwete kutora mishonga pa:
- bradycardia (kwemwoyo Me anorova 50 paminiti);
- SSS;
- nhaka galactose malabsorption kana kusashivirirana (shuga)
- Lactase kushaikwa;
- yakawedzera aikanganiswa zvinoriumba nzira;
- vana uye kuyaruka pasi pemakore ruzhinji.
Zvokungwarira ramakanzi mushonga ari chinouraya chokutambudzika kana zvakakomba renal kukundikana, varwere vari pasi hemodialysis, kwazvo chiropa kukundikana.
Mahwendefa "Fiziotenz": zvairatidza kuti kushandiswa, ongororo, mirayiridzo inokosha
Primary nechirwere, umo vanachiremba mishonga iri neBP. Zvinofanira kurangarirwa kuti panguva kurapa vanofanira kuita hurongwa richiona mamiriro BP, ECG uye kwemwoyo. Kana uchida kukanzura mishonga, ipapo ichi chinofanira kuitwa zvishoma nezvishoma.
The chigadzirwa hazvirevi kukanganisa kukwanisa kudzinga uye zvifambiso zvigadziriswe. Zvisinei, kuti idzidziso "Fiziotenz" (murefu uchapupu hunoratidza kuti izvozvo) vaifanira kutora nokungwarira nokuti kunogona kukonzera dzungu uye hope. Izvi zvinofanira kufungwa vanhu vaiita ngozi, rinoda kugara yevasungwa, mabasa.
Storage mamiriro, analogs uye mutengo
Mahwendefa zvinofanira kuchengetwa panzvimbo vana havagoni kusvika. Pasi nemitemo okuchengetera (tembiricha kusvika 25 ° C, iyo yakaoma rima panzvimbo) zvinodhaka haangaregi kurasikirwa pharmacological ehupfumi dzavo, kwemakore maviri. Buy mishonga "Fiziotenz" (wongororo ngaadarowo) zvinogoneka pamusoro mushonga mu Pharmacies. Price kavha mahwendefa (0.2 MG) ndiyo 275 rubles. Kana mishonga panguva chemishonga vamwe chikonzero haana, zvakakodzera kutarisa vezera: "Cynthia," "Moksoniteks", "Moxonidine", "Moksogammu".
Reviews kugadzirira "Fiziotenz"
Varwere vakawanda vanotaura pamusoro mushonga sechinhu nzira inobudirira yepamusoro. Vanhu vanoti kuushandisa kwemakore, mushonga lowers BP zvakanaka, pasina nemishonga. Vamwe vanotaura zvinokanganiswa kudhura Mahwendefa "Fiziotenz". Reviews zvinoratidza kugarisana zvakanaka nevamwe nzira vane chirwere cheBP mishonga.
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