Utano, Gadziriro
'Betalok' mirayiridzo kushandiswa
"Betalok" mirayiridzo Chinyorwa rinotsanangura sezvo mushonga kungova pharmacological boka beta1-adrenoceptor mhandu. The chikuru vanoshingaira wemafuta zvinodhaka ndiko metoprolol tartrate. Zvinonzi zvinoberekwa vagadziri muchimiro mahwendefa mashekeri 100 milligrams, vari mumapepa mupurasitiki hombodo dzemvura zvidimbu 100 nerimwe.
"Metoprolol" ane pharmacological ehupfumi, inobva mano zvinodhaka kupa antihypertensive uye Anti-anginal chiito. The mushonga unoshanda mukuderedza kwemwoyo, myocardial contractility uye excitability, kunosimudzirawo deceleration pezvakaitwa AV-conduction. Kugadzirira "Betalok" mirayiridzo Chinyorwa anorondedzera kuyamura zvinoderedza cardiac Vhoriyamu uye okisijeni ukapisa nokuda myocardium. "Metoprolol" anokwanisa kuderedza catecholamines pa masero kukanganisa kwavo pamusoro murwere mwoyo munguva psycho-mumuviri mupfungwa. The mushonga une hypotensive zvazviri pakudzikamisa pashure pemavhiki maviri kurapwa. "Metoprolol" rinoratidza efficacy yakakwana pakurapa navanopinda chakarondedzera zvemwoyo, pakati rinogona kuzivikanwa myocardial infarction, coronary tsinga chirwere, arrhythmias pamusoro siyana, unoshanda senzira prophylactic mumiririri kudzivirira dzokororo kurwiswa mwoyo.
Pharmacokinetic ehupfumi "Betalok" zvinodhaka mirayiridzo kushandisa zvinotsanangurwa nenzira iyi. Pamusoro nokugamuchira substantially vose mushonga munguva pfupi uye wefodya kubva nemudumbu, ayo kunonyanyisa wevasungwa munguva plasma runowanikwa mukati maawa imwe kana maviri. The mushonga unogona kukurumidza rinoita ari chiropa, nokudaro yakabereka metabolites vane chinenge hapana basa mhosva chero muviri miviri. The hafu-upenyu zvinodhaka zvinoriumba iri anenge matatu kana mana maawa, uye kushanda haachinji kuti nguva yose kurapwa. Excretion pamusoro metoprolol anogadzirwa itsvo - anopfuura 95% of dose yamarudzi, sezvamakaropafadzwa hapana zvinopfuura zvitatu muzana inenge yabudiswa kuchinja.
"Betalok" muperekedzi anokurudzira kuti vanenge zvinotevera zvirwere nokuti kurapa BP, sezvo muviri mumiririri rinoshandiswa kudzivirira kurohwa. A mushonga kuratidzwa vanenge cardiac arrhythmias, uyewo yechipiri kudzivirira zvinodiwa pashure kutambura cardio-vascular hurongwa.
The chipimo chemushonga zvaiitwa zvinodhaka "Betalok" mirayiridzo Chinyorwa anokurudzira kuti iwe dzishandise ichi. Avhareji dose zvinodhaka kaviri pazuva iri negashiro milligrams 100 pazuva. Mune zvimwe zviitiko, mirayiridzo iroro mukana zvishoma nezvishoma yakawedzera dose kaviri. Kana mushonga unoshandiswa nomutsinga, chete dose zvichisiyana 2 kusvika 5 MG. Kana iyi haina kubudirira zvinozoita, kugadzirira inogona kupiwa kakawanda pashure maminitsi 5.
The chipimo chemushonga zvaiitwa anofanira kufunga kuti pokushandisa kunonyanyisa dose zvinodhaka riri 400 MG pazuva.
Kana kugamuchira mapiritsi "Betalok" anogona kukonzera marwadzo kubva siyana enyika muviri. Pachikamu yavo hwakadzama uye tsanangudzo zviratidzo anopiwa mune mirayiridzo kushandiswa kwezvinodhaka.
Contraindications kugamuchira mishonga yakasiyana maererano mhando uye hunhu kuyerera blockade zvemwoyo conductivity, hypotension, cardiogenic kuvhunduka nezvimwe zvirwere. Contraindicated Kugamuchirwa kana murwere ane hypersensitivity kune yenhengo dzayo. Regai kutora zvinodhaka panguva yepamuviri uye achiyamwa.
Nokungwarira yokunyanyisa anofanira akaswedera kushandisa zvinodhaka nevarwere vane COPD,
cheshuga, chirwere Raynaud vake.
Zvokurega mishonga yakarumbidza zvishoma nezvishoma, izvi zvinofanira kugara mazuva anenge gumi.
The mushonga ane vanoverengeka dzinokosha modes kuita, kuburikidza tichibatanidza pamwe nezvimwe zvinodhaka. ruzivo urwu uchida inowanikwa mune mirayiridzo kushandiswa.
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