Utano, Gadziriro
"Omeprazole" kana "Ultop" - inova nani? Description zvinodhaka, zviratidzo uye contraindications, mitengo
Mabatirwo maronda maronda mudumbu mucosa kana zvomudumbu turakiti zvavo - kunzwisisa uye dzakareba muitiro. Izvi imhaka kwete chete kune chokwadi kuti hydrochloric acid, chikamu gastric muto, inowedzera zvishoma nezvishoma mucosa kuremara, digesting pachake munyama, asi kuwadzana pamberi chirwere Helicobacter pylori microorganism. Kuitira kudzivirira pakuwedzera kuremara uye aivabatsira kukurumidza kupora murwere, vanachiremba akarayira "omeprazole" kana "Ultop". Ndezvipi zviri nani, tichakurukura munyaya ino.
mashandiro chiito
Pasinei nokuti zvinodhaka akasiyana zita, zvinoshingaira pazvokudya kwavari zvakafanana - omeprazole. Anorapa uye mushonga uyu?
Maererano makemikari unhu fuma iri kushanda insoluble nemvura, asi chaizvo soluble mu panyaya iyi kana methanol.
In kurapwa tsika, omeprazole rinoshandiswa Zvinoumba zvinodhaka zvakasiyana-siyana, kusanganisira mubatanidzwa, sevamiririri kuti kurapwa nemaronda. "Omeprazole" kana "Ultop" - inova nani? Kakawanda ini kuzvibvunza mubvunzo uyu, varwere uye vanachiremba.
The mashandiro chiito kwakavakirwa chinovhiringidza kunzi hwepurotoni pombi - dzakananga chokufambisa mapuroteni iri muchitokisi Kamudzira pamusoro secretory masero ari mudumbu. Akaroromesawo kubvuma rehydrogen ions vari cytoplasm masero secretory kwakadaro ungaderedza wakabura inobereka hydrochloric asidhi uye acidity pamusoro gastric muto kunodzikira, iyo inosvitsa zvinoderedza zvinyama kuparadza uye anofarira wakakurumidza nokuporesa nemaronda.
Pharmacokinetics
Omeprazole zvinobudirira kuchititadzisa zvose dzinovhurika uye basal kugadzirwa hydrochloric acid, panguva iyoyo dose kuzvimiririra kushanda. Kana rimwe nomumukanwa kwokubatsira 20 MG "omeprazole" kana mabiko dose "Ultop" gadziriro - 20 MG, acidity kuderera ari kuchengetwa mukati awa rokutanga, sezvo mushonga uri nokukurumidza uye tsime woga kubva intestinal lumen uye anopinda systemic kutenderera.
Kunyange zvazvo hafu-upenyu vanoshingaira mumiririri Formulations iri maawa anenge maviri, chinovhiringidza ari kudhindwa hydrochloric asidhi ari kuchengetwa mukati memazuva pashure chete dose.
Omeprazole mudungwe munzira partitioned nokuda chiropa uye biliary turakiti mucous Kamudzira mudumbu, kushanda asingadi zvinopfuura ropa-uropi chipingamupinyi uye anosungirwa chose kuti mapuroteni eplasma. The mwero tichisunga pamwe yokupedzisira inogona kusvika 90-95%.
Excretion pamusoro omeprazole rinoitwa kunyanya weti, pamwe vanenge 60-77% iri yabudiswa muchimiro metabolites akadai gidroksiomeprazol uye carboxylic acid. Vakawanda zvichizoita verlauf kuratidza chinenge hapana antisecretory basa, kunze sulfonomeprazola. The yasara muviri chikamu zvinodhaka fuma anoratidzwa ne nemudumbu ari bile uye faeces.
Special ngwariro vanofanira pharmacokinetics kuti omeprazole pavarwere vane hepatic insufficiency. Akaroromesawo muviri zvinodhaka zvasvika vaifanira bioavailability uye hafu-upenyu nguva kuripo maawa matatu. In varwere chisingaperi renal insufficiency DZEMUNHU DZINODZORA excretion pamusoro metabolites ose omeprazole maererano wokunatswa plasma creatinine.
zvairatidza
Zvinodhaka "omeprazole" uye "Ultop" kwakaratidza kuti kushandiswa pakurapa peptic nemaronda ari zvomudumbu turakiti, hyperacidity inoti (kusanganisira gastritis), Zollinger-Ellison urwere, postoperative mamiriro ezvinhu reflux chirwere. mishonga iyi inogona kurumbidzwa kuti pakurapa asiri urikanwi dyspepsia Genesisi mukurapa yematambudziko akakonzerwa non-steroidal kurapa protivovospalitelnymim zvinodhaka (analgesics, antipyretic), uyewo nokuda pakurapa nyore chirungurira kuti kunoitika anopfuura 2 nguva pavhiki.
Pasinei mirayiridzo iri zvairatidza kuti kushandiswa zvinodhaka "Omeprazole" kuti ichibata chinodhaka, anoziva chete yakarovedzwa mukoti. Saka, kana uchifunga kurwara, kubva nemudumbu, unofanira kuenda kukiriniki uye kwete kuzvinzwira medicate.
Contraindications
All marudzi ose chinodhaka, kusanganisira mapiritsi "Omeprazole" iri contraindicated pamberi varwere hypersensitivity kuti mushonga, uyewo vana. Kuderedza secretory kushanda mudumbu kana hypoacid inoti uye atrophic gastritis ariwo contraindication kwokugadzwa omeprazole.
nemishonga
Pamusoro mushonga "Omeprazole" uye "Ultop" wongororo vanoti, nokuderedza asidhi-achiumba kushanda mudumbu, kubva nemudumbu zvichida kuti kupatira, bloating, kupatira, kurutsa uye kurwadziwa epigastric nharaunda. Kashoma vakachengeta candidiasis, muromo yakaoma, kana kuvandudzwa atrophic hypoacid gastritis, polyposis pamusoro ura.
Kubva tsinga (kutsinga dzinouya chiyamuro), unogona kuona nemusoro, zvakawanda zvive, kufunganya uye manzwiro kuzvidya mwoyo uye zvinetso mupfungwa. Zvinokwanisika kuti kwaita zvinetso zviri kutarisana basa kuti anogona kuva zvechigarire.
Sema kwomusikirwo omeprazole hadziwanzowaniki. Situation kungaita mikoko, kuvaviwa. With yakaderera maitikiro manotsi gladomyshechnyh Árbol spasm sero kukura angioedema ane mberi kuchiita mhando anaphylactic siyana uye kukura nehana sosotoyaniya. Casuistically akaona kukura gynecomastia, pakuonekwa marwadzo ari pachipfuva.
Dosing
"Omeprazole" tora usina chawadya nemvura. Mune chikamu chaiye varwere vanogona kunetseka pakuparadza capsules zvinodhaka. Muchiitiko chino, Zvinokurudzirwa kuvhura Kamudzira uye zviri mariri kubva slurry agadzire mvura-inobva. ari kumisa anofanira kutora kanenge hafu yeawa pashure kubika. The daily chipimo chemushonga, imwe dose, uyewo nzira zvinodhaka mishonga unogadza chiremba.
Zviri kushanda munyika nhumbu uye uchiyamwisa
Data pamusoro kuchengeteka omeprazole vakadzi vane pamuviri havana. The mushonga fuma kungaratidzwa nezvikonzero zvoutano. Category migumisiro pamusoro azvarwa hazvina vasarudzirwa.
Kana pane kudikanwa kugadzwa omeprazole panguva achiyamwa nguva, ipapo pakurapa yokupedzisira ndiko kuramba, sezvo mushonga anogona kupinda mu zamu mukaka.
Drug kwavatori
Se "omeprazole" uye "Ultop" kuderedza bioavailability mishonga, iyo Absorção de Água iyo kunoenderana acidity ose gastric muto. Uyewo kuchititadzisa kusunungurwa zvinodhaka izvo muviri ari chiropa.
Kugadzirira chena injectable mhinduro kubva omeprazole kungashandiswa kwemaawa 12 akapa kushandiswa vasiri yavaibvisa chloride mhinduro sechinhu solvent uye kwemaawa anoverengeka pashure kugadzirira kana kushandiswa senzira solvent dextrose mhinduro. Nevamwe zvingaitwa omeprazole haienderani.
With concomitant kurapika "Warfarin" rinofanira kuongororwa daily anticoagulant nhanho mu plasma kana nenguva netsika kuongorora zviri prothrombin nguva.
chepfu uye ovhadhozi kurapwa
Symptomatology omeprazole ovhadhozi kunoratidzwa sezvo muromo yakaoma, dzungu, nomusoro uye vasanyatsoona. Kana muchetura zvinobvira kuvhiringidzika, panowanikwa nehope, palpitations, Flushing manyawi.
chepfu symptomatic kurapwa zvainanga sei kuti zvikuru nokukurumidza kubviswa pakati zvinodhaka mumuviri. A wakananga mushonga haizivikanwi. Nokuda mukuru mwero tichisunga kuti mapuroteni eplasma, kushandiswa dialysis detoxification nzira seisingashandi.
Zvokungwarira
Sezvo mishonga inoshandiswa kurapa maronda maronda mudumbu uye duodenum, ndiko etiological mumiririri Helicobacter pylori chirwere, Zvinokurudzirwa kuti yokupedza zvigare concomitant kwokubatsira antibacterial zvinodhaka.
Asati atanga kushandisa zvinodhaka pane murwere unofanira kuramba nyanyisa neoplastic zvirwere nemudumbu, sezvo kugadzwa "omeprazole" kungavanza zviratidzo zvirwere izvi uye kuchidzivisa mangwanani kuongorora chirwere. Zvakakosha kubvisa parasitic zvirwere, uyewo kuongorora dzichipfekeka vachikwanisa chiropa uye neitsvo.
"Omeprazole" kana "Ultop" - inova nani?
A mhinduro yakajeka yomubvunzo uyu kwakaoma, nokuti basa fuma, uye pose ndiyo omeprazole. Ngatimboonai chimiro kusunungurwa zvinodhaka "Ultop". Capsules anogadzirwa mune chipimo chemushonga 10, 20 uye 40 MG, uyewo lyophilized upfu (40 MG imwe chinu) achigadzirira jekiseni mhinduro.
"Omeprazole" anoratidzwa pamusoro mishonga pamusika muchimiro capsules 10, 20 uye 40 MG kuti omeprazole imwe Kamudzira, uyewo lyophilized upfu (40 MG imwe chinu) achigadzirira jekiseni mhinduro. -oma-kuomeswa upfu pamwe solvent kuri kuwanikwa mune chete pasuru. Uyezve, mushonga inogona kutengwa muchimiro sachets (mumasaga pamwe madota) achigadzirira nomumukanwa kuturika. Kashoma ane "omeprazole" Mahwendefa (pellets) pamwe chete zviri zvinodhaka fuma.
Kana wongororo nezvezvinodhaka izvi, vava akanaka, sezvo omeprazole inzira inobudirira chinodhaka kuti akazoita secretory basa mudumbu. The mushonga unoshanda kuitira kuti kunyange vanachiremba vari kubvunza, "chii nani omeprazole" Zvisinei, maonero akasiyana pavarwere. Kazhinji vakasiiwa zvinodhaka "Ultop" wongororo vanoti nezvemavambo kupatirwa pashure ingestion, nomusoro uye svoto.
Mari zvinodhaka
Zvechokwadi, mari zvinodhaka kuchaenderana kwete chete pane chemishonga samambure yavanofanira dzinotengeswa, asiwo chinhambo kubva kuchipatara chemishonga uye, chokwadi, kubva zvinodhaka mugadziri. The mushonga "Ultop 'mutengo neeSultan kubva 212 kusvika 360 rubles muzana rongedza. Kwokupedzisira mutengo kunobva dose uye uwandu capsules por bhokisi. The mushonga "Omeprazole" mutengo iri avhareji kubva 80 kusvika 140 rubles. The mutengo inobvawo pamusoro dose uye uwandu capsules por bhokisi.
mhedziso
Chete chiremba anofanira mishonga "Omeprazole" kana "Ultop". Kuti akanakisisa zvinodhaka izvi, anoziva hwakakwana munhu, uye sarudzo kwayo kunofanira inobva zvairatidza uye murwere ezvinhu. Zvinofanira kurangarirwa kuti kazhinji inokosha chinokonzera pakusarudzwa zvinodhaka ndiko wayo mutengo.
Varwere vanofanira kuteerera "omeprazole", riri yekudyidzana kudzika mutengo pane analogue "ultop". Vaya vanoda mari zvikuru, vanogona kutarisira analogues zvinodhaka. Pasinei hwaikosha dzakawanda "Ultop" chinodhaka mutengo aigona kupembedza ukuru wokunatswa chinodhaka, uyewo zvichibvira mamwe kugadzirira modulating chirungiso pacharo.
Chero zvakanga nguva dzose zvakakodzera kuyeuka yendarama ushe: regai kuzvidzora medicate. Early chirwere - kiyi akabudirira kurapwa!
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