UtanoGadziriro

"Antabuse" mapiritsi. Reviews, mutengo gwaro

It akadana udhakwa chirwere kunoratidzwa muropa panyaya iyi pamwe mumuviri uye havakwanisi payo. mhando iyi kushungurudzwa. In mamiriro ichi, kurasikirwa kudzora uwandu akadhakwa doro kunowedzera achishivirira pazviri (kuzadzisa kugutsikana doro nguva kuwedzera dose) uye kushaya chirwere kunoitika, chinobata nhengo dzomukati uye kuoneka ndangariro dzakaipa.

Varwere kutambura udhakwa, vanonzi zvidhakwa. Kubata chirwere chinofanira mupfungwa nomumuviri. Kakawanda, vanachiremba akarayira zvinodhaka izvi kuvanhu "Antabuse". Mirayiridzo kushandiswa, mitengo mishonga, zvokurapa wongororo vanoonekwa pazasi.

Apex, chimiro, uye mamiriro tsananguro

In chii vanoumba zvinodhaka anotengeswa "Antabuse"? Testimonials dzinoshuma kuti yakadaro mushonga inogona kutengwa muchimiro chena, kumativi effervescent mahwendefa. Vane sandara, beveled unopinza, pangozi uye nokuyera «CD» uye «C» kumativi akasiyana ose ngozi.

The Zvinoumba mishonga iyi anosanganisira disulfiram. Kunze kwayo, kugadzirira rine zviyo starch, povidone, yavaibvisa hydrogencarbonate, tartaric acid, colloidal nesilicon dioxide, talc, microcrystalline cellulose uye magnesium stearate.

Mahwendefa "Antabuse" akaisa mupurasitiki midziyo uye packs it makadhibhokisi.

pharmacodynamic unhu

Chii chinodhaka "Antabuse"? Manual rinoti izvi zvinoreva antialcoholic. It kuchititadzisa acetaldehyde dehydrogenase, iyo rinobatanidzwa muviri panyaya iyi. Kunonotsa kwayo oxidation kwacho kunokonzera kuunganidza doro uye pave simba kudhaka, ichiteverwa rinorema manzwiro ari throbbing kurwadziwa uye ruzha mumusoro, tachycardia, palpitation, zvinoderedza BP, kuda kurutsa, madzerere uye kurutsa.

Maererano nenyanzvi, zvisingafadzi zviratidzo izvi zvinobatsira kuti pave vakaumbwa dzepanguva mukupandukira doro.

pharmacokinetic ehupfumi

ari Absorção de Água kuti "Antabuse" chinodhaka sei? Manual kunoratidza kuti mushonga wefodya nokuda 70-80%. Iye zvikuru soluble mune lipids uye uderedze kuunganidza ari mafuta dhepoti.

The kushingaira pafuma pomutumwa yava kwazvo rinoita, zvichiguma vakachinja metabolite - methyl Ester dietiltiokarbaminovoy acid. kuwanda Parainge ropa vakatsunga pashure 4 h. Kunyange zvazvo basa pachinhu acetaldehyde dehydrogenase ari kuchengetwa chete pashure pemazuva matatu.

The hafu-upenyu zvinodhaka ndiko maawa 10. Uyezve, kwayakaita pamusoro aldehyde dehydrogenase anoramba yakareba. Naizvozvo, pashure kudzimwa pakati zvinokonzerwa mahwendefa zvinochengetwa kwenguva mamwe mazuva 7-14.

The mushonga rinowanikwa weti, uye pamwe kuburikidza muura pamwe patinofemera kunze mhepo.

umboo

Mune zvimwe zviitiko, inonyatsobudirira zvinodhaka achiita "Antabuse"? Reviews akashuma kuti chivako ichi rinoshandiswa chaizvo kudzivisa kuitazve pakurapa doro nedoro uye chidhakwa.

Contraindications

Kana iwe haufaniri kutora "Antabuse" piritsi? Guest vanamazvikokota vanoti vaiona mushonga harifaniri ushandiswe kana:

  • yemaziso;
  • neuritis of optic uye auditory tsinga;
  • pulmonary tiibhii;
  • mwoyo uye vascular zvirwere (semuenzaniso, post-infarction rinoti, akaratidza cardiosclerosis, atherosclerosis pamusoro chepfungwa midziyo, vane chirwere cheBP chirwere, kutsemuka aneurysm);
  • polyneuritis chipi mavambo;
  • chirwere cheshuga;
  • emphysema, Árbol asima;
  • thyrotoxicosis;
  • mupfungwa kurwara, pfari uye epileptiform chirwere;
  • akaipa mota;
  • chakakomba hepatic uye renal kukundikana;
  • zvirwere hematopoiesis;
  • exacerbation pamusoro peptic urikanwi chirwere;
  • pamuviri;
  • hypersensitivity.

Onawo kuti zvinodhaka izvi hama contraindications:

  • makore 60;
  • migumisiro sitiroko pamwe residual zviratidzo;
  • peptic urikanwi (kusanganisira rekukangamwirwa);
  • precipitates munhu psychosis.

Drug "Antabuse": mirayiridzo kushandiswa

Anti-doro piritsi mutengo akanyorwa pakuguma nyaya. Vanofanira kutora mavo ½ kare zvazvichanyungudutswa girazi remvura.

Kazhinji, vanachiremba akarayira 200-500 MG zvinodhaka kamwe kana kaviri pazuva. Pashure pemazuva 7, iva nechokwadi kuti kupedza disulfiram-doro bvunzo. In kufanana negashiro 500 MG ose medicament murwere zvinwiwa 20-30 ml vodka. Kana kuita simba, ipapo kuwedzera dose doro kusvika 20 Rine mamiririta.

bvunzo iyi inodzokororwa kakawanda. Papera ballroom ushandiswe Nokuraramisa chipimo chemushonga kuti 200 MG zuva nezuva kwemakore 1-3.

nenjodzi

Mahwendefa "Antabuse", iro ratings dzinoturwa pazasi kungaita zvinotevera nemishonga:

  • chiropa, asthenia, simbi kuravira mumuromo;
  • cutaneous kuratidzwa, polyneuritis tsoka;
  • kurasikirwa ndangariro, pfungwa kuzvimba, nomusoro;
  • myocardial infarction, cardiac arrhythmias;
  • kufema kukundikana, zvemwoyo dhirika;
  • optic neuritis, chepfungwa thrombosis midziyo;
  • psychoses, angina.

Medicament "Antabuse": wongororo kuvarapi uye mutengo

Mari mahwendefa Anti-doro anenge 450-600 rubles (zvichienderana dose uye uwandu pa rongedza).

Vanachiremba vane mishonga ine mushonga wakadaro, pakarepo akayambirwa yematambudziko chakakomba chinogona kuitika mune murwere necheseri zvichakutorera. Naizvozvo zvachose wairambidza kubata pachako kana zvakavanzika kubva murwere.

Zvinofanira kucherechedzwa kuti nyanzvi dzakawanda dzinobvuma kuti zvinodhaka vanobudirira kuti vasaziva nehavi doro, kwete. Uye nzira iyi haisi kurapa. Rinongotaura anosimudzira yakagadzikana kanganwiro.

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