UtanoGadziriro

The mushonga "Tamsulosin": mirayiridzo kushandiswa, mutengo, wongororo uye analogues

"Tamsulosin" antidizuricescoe ndiwo mushonga chiito uye rinoshandiswa senzira symptomatic Urinary modulator kwacho Urological zvirwere zvinokonzerwa sero-akaipa prostate anomera hunhu. The Zvakaitwa mashandiro kunoratidzwa zvishoma nezvishoma kuderera kuchinyanya munyika anotsvedzerera tsandanyama kweprostate, uyewo kutandara ari dundira mutsipa. Uyezve, pane kusarudza ichivharira urethral Alpha 1a-adrenretseptorov, zvichiguma minimization migumisiro vakachengeta mhingaidzo - munhu wechisikigo mugumisiro pokumuka adenomas.

Pharmacological zviri "Tamsulosin"

Absorção de Água zvinodhaka unorapa mune nemudumbu inogona kusvika 100%. Experimentally akasimbisa kuti Absorção de Água ichiwedzerwa apo kutora capsules pakarepo pashure zvokudya. The mwero kuitwa Proportional kusvikira nguva yakapfuura kubva kudyiwa zvinodhaka (i.e., pane Linear kinetics). Yepamusoro wevasungwa zviri reactants mu plasma runowanikwa pashure maawa matanhatu (kuroora dose 400 MG). Zvisinei, nguva nenguva ino dzingasiyana zvichienderana nemakore murwere.

Zvinonzi kuzivikanwa kuti mabiko panguva Chokwadi mazuva mashanu, wevasungwa pakati zvinoumba mu plasma inowedzerawo kubudikidza 60-70%. Tamsulosin hydrochloride zvakakwana zvishoma nezvishoma anopinda metabolic pezvakaitwa: uptake pamwe paumbwe akatsiga metabolites iyo vane yakakwirira selectivity nokuda Arifa 1a-adrenoceptor.

zvairatidza

The mushonga "Tamsulosin" mirayiridzo Chinyorwa classifies okutenderera nokuda pakurapa prostatic hyperplasia isiri yekenza, zvikuru symptomatic (adenoma, dysuria, uye vamwe ezasi yokubereka turakiti chirwere).

Sezvo kurapwa zveBhaibheri havana kwakaratidza chero dzinonetsa zvinoitwa zvimwe zvinhu zviri vakati boka mishonga, saka hapana rairambidzwa kushanda "tamsulosin" webetsero tiwedzere pamwe navanachiremba ichivharira zvokusarudza Alpha-1a adrenergic Kanotokonya.

Recommended chipimo chemushonga uye nzira chourongwa

Kushaya hypotensive maturo - anozivikanwa chepfungwa zvinodhaka "Tamsulosin". Mirayiridzo yokushandisa rinoti kuti kudiwa dose kusarudzwa oga haisi - zvakakwana nomuromo raitongwa 400 micrograms zvinodhaka pashure pokudya kwemangwanani (2 capsules / mahwendefa yairema MG 200 neimwe, kana 1 Kamudzira / piritsi yairema 400 MG). Uyezve, mwero iri zuva hakufaniri kugadziriswa, kunyange kana murwere kuchengetwa zviduku zvarakasiya ari itsvo kana chiropa. Kunyange zvakadaro, pakutanga kuchirapa Chokwadi anofanira pakurukurwa chaiyo chirwere kuti kudzivirira kubata kenza yeprostate. Uyewo panguva dzose panguva kurapwa vari fanira rectal kuzviongorora.

Capsules uye mahwendefa "tamsulosin" haafaniri kutsenga - kutyora hamvuropu kunogona kukanganisa kusunungurwa mwero yezviri reagents. Pakarepo mushure kutora mushonga inokurudzirwa kunwa mvura. Zvinonzi zvaisambobvumirwa kushandisa "Tamsulosin" iri supine chinzvimbo.

Huripo zvausingakwanisi uye contraindications

The mushonga "Tamsulosin", mutengo iyo, zvichienderana mugadziri uye kavha zvinogona, yemakomo 400-1700 rubles, akagadzirirwa chete varume. Saka, kuongorora migumisiro ayo pamusoro azvarwa vasina inoitwa panguva yepamuviri. chete mushonga inowaniswa chinyorero data, kureva, zvokuongorora kuti "prostatic hyperplasia isiri yekenza" anofanira ari kuongorora (ane fanira pre-muedzo kenza).

Pakati contra - hypersensitivity kuti "Tamsulosin" chinodhaka (User chikumbiro ine ndandanda zvose hwebetsero reagents). Hazvina kunaka kushandisa kuti akati mumiririri kuti orthostatic hypotension uye chisingaperi nezvirwere chiropa kana itsvo (mu Pakadaro, chiremba anofanira kufungidzira uchabatsirwa mashandisiro "tamsulosin" uye kuona kukura kwakaita zvingangoitwa migumisiro muviri kosi).

With nguva kugamuchira bvumidzwa chiedza dzungu, dzimwe nguva chakatsiva semiconscious mamiriro. Vatyairi motokari uye vashandi, ane mabasa nyanzvi inosanganisira ngozi kukuvara, vanofanira kuchengeta kungwarira kunyanyisa pakushandisa nefuma.

nemishonga

Kufanana mimwe zvinodhaka, pane marwadzo uye zvinodhaka "Tamsulosin" (mutengo utano avanhu zvakakwirira, uye neutachiona zviri zviduku, saka kuti nenjodzi sechinhu chinokosha kusava hazvina zvakakodzera).

In kufanana kupodzwa zvinogona kutora nzvimbo:

  • nomusoro;
  • kutsamwa ganda;
  • ya manyoka;
  • cardiac arrhythmias;
  • pelvic marwadzo.

"Tamsulosin" Dzimwe nguva, analogues zvacho zvikuru pa pamusika, zvichiita kushaya hope varwere kana, Ukuwo, kunyanya nehope. Mune zvisingawanzoitiki kacho - kwekanguva kutyora cheya uye kwakaderera potency.

Ovhadhozi, kuonekwa uye neutralization

Zviratidzo ovhadhozi, razova migumisiro zvinodhaka riri "Tamsulosin" (mirayiridzo kushandisa zvinonyevera iyi), zvinogona ritaurwe rikwanise hypotension. Uye kunyange mukana wokuti muchiitiko ichi yakaderera zvikuru, kuti algorithm kubatsira zvakadaro akaita:

  • pakarepo kupa murwere chinjikira nechinzvimbo;
  • kana zvakafanira, vaite kunzwisisa zviyero zvainanga ari normalization pakati kumwoyo kwemuviri;
  • kuti asimbise mashandiro anoita itsvo (kubatana midziyo kubata ropa yokuzvinatsa dzisingashandi nokuti rinoita chirungiso anonyatsorayiridzwa chokuita yeplasma yeimwe);
  • kukonzera manyoka murwere kuti kurega zvimwe Absorção de Água pamusoro reactants (uyewo wechokwadi gastric lavage pamwe yakafanana kushandisa laxatives);
  • pasina simba rinomutsa yokuchinja kushandisa mishonga inotokonya kweropa.

Drug kwavatori: yezvakaita siyana

"Warfarin" uye "Diclofenac" qualitatively kukanganisa goho kumhanya "Tamsulosin" chinodhaka muviri (zvinodhaka mutengo yakawanda, asi mugumisiro zviripo). Zvisinei, kwenguva yakareba zvaanorumbidza maererano vagari kushandisa zvinodhaka izvi muchipatara isina kuitwa, sezvo zvakaguma kungwarira akanyanyisa inokurudzirwa. "Atenolol" uye "Enalapril" asingadi kushamwaridzana akati zvinhu, "cimetidine" anosimudzira pfungwa "tamsulosin" plasma, uye "Furosemide" anopa zvachose zvinake.

Muitiro BP kushatiriswa yaunodya pamusoro medicament anogona huchawedzerwa nokuda pamunhu yaizoshanda panguva kushandisa mamwe Alpha-1a adrenoblokatorovv kana diuretics uye dzokutindivadza. Chinokosha zvainoita pharmacological kinetics chokuzvisarudzira zvikamu zviduku "Diazepam" uye "chlormadinone" ne kugadzirira "Tamsulosin" mirayiridzo Chinyorwa (mutengo pamusoro nzira -. 500-1400 NZD) haisi kunorondedzerwa.

Storage mamiriro uye sherefu upenyu

On kuchengetera zvinhu zvinodhaka "Tamsulosin" muperekedzi inoti zvinotevera:

  • yakachengeteka tembiricha Range - 15-25 Celsius;
  • optimum mwando - 70%.

Chinodiwa kuchengetera zvinhu chepakutanga kavha (panzvimbo dzisingambosvikiki vana, iro tsime kudzivirirwa zvakananga chezuva).

Kana pfungwa dzose mirairo mugadziri hunovimbisa kuti mishonga chaizvoizvo "Tamsulosin" vachange kuregeredza makore maviri kubva kwayo kusunungurwa.

Drug analogues "Tamsulosin"

Ndandanda "Paarismängud" anomirirwa nemapoka maviri zvinodhaka. Boka rokutanga zvinosanganisira mishonga, zvakafanana, wechipiri - isingawanzowanikwi dzaishandiswa mazita.

Public mari:

  • "Omnic" (mu epakutanga - Omnic), mugadziri - Netherlands, vasunungurwe chimiro - mapiritsi / capsules 10/30 zvidimbu por rongedza, mutengo siyana - 380-1700 rubles.
  • "Proflosin" (Proflosin), Germany, Maronda akasiyana pamusoro capsules 30, nokukosha mutengo - 500 rubles.
  • "Sonizin" (Sonizin), Kunyika kwayakabva - Romania, chiyereso pasuru 10 kana 30 capsules, avhareji yemari - rubles 450.

Mamwe trademarks uye kutengeserana mazita zvinodhaka "Tamsulosin" (analogs kuti vari ishoma kana kusunungura siyana akatowana kubva production):

  • "Omsulozin" (Omsulosin), India, capsules 0,4 MG (30 hrs.) Price neeSultan kubva 350 kusvika 550 rubles.
  • "Tamsulosin-din email" (Tamsulosin-din email), "Tamari-Actavis" chigadzirwa kambani, Greece, chimiro kavha uye mutengo kwakafanana muzvirevo nyaya.
  • "Tamsulosin-kutadzisa" ( "understudy" kuramba kusunungurwa chazvo), kurimwa mutsetse vakagara Russia, mapiritsi 400 MG, mutengo - vanenge 300-360 rubles.

"Tamsulosin": wongororo vanachiremba uye varwere

Medical kurapa pamwe kwezvinodhaka izvi kazhinji kubudirira uye runoratidzwa munzira regression mashoko kuri vasiri akaipa yeprostate anomera.

Mushure anenge 90 mazuva zviratidzo aiitwa muna 2 nguva yokutanga kuchinja kuoneka vakatobatana pasika mazuva 14-21. Panopera zviratidzo mapopoma indekisi ne 75% (mu tichienzanisa kutanga danho), iro zvechokwadi zvinogamuchirika mugumisiro.

Beautiful tolerability "Tamsulosin" (gwaro mutengo uye rakajairika mishonga Generic vanopiwa pamusoro) zvinoita nyore chaizvo kushandisa kana rakavapa varwere mishonga. Zvisinei, kuti vabudirire kunonyanyisa zvingaitika nefuma iri kushomeka, Zvinokurudzirwa kuti pamunhu yaizoshanda panguva kurapa nevamwe nzira uye mishonga zvigadzirwa.

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