Utano, Gadziriro
"Buspirone": nhoroondo, mirayiridzo kushandiswa, analogs
"Buspirone" rinoreva mari kuti kuva nezvahunoita tsinga. Hazvina anxiolytic, zvakagadzirirwa kubvisa mwoyo uye kutya, normalization hope, kuvandudza zvakanaka pamberi neurosis. Mahwendefa "Buspirone" mamwe contraindications, uye zvinogona kukonzera marwadzo.
Murwiyo uye chimiro "Buspirone" chinodhaka
The mushonga inowanika Hwendefa muchimiro panguva chipimo chemushonga 5, 10 uye 20 MG. The rinoita mushonga fuma - buspirone. Ebetsero zvinhu zvinosanganisira potassium hydroxide, chibage starch, magnesium stearate.
Pharmacological migumisiro
Zvakaitwa zvinodhaka kunyaradza, anxiolytic. The mushonga anobvisa zviratidzo nokutya vegetative uye utano hwepfungwa. zvinoreva mashandiro chiito haina chose kunzwisiswa, asi inozivikanwa kuti "Buspirone" rakasiyana benzodiazepines uye zvimwe zvinodhaka anxiolytic kushanda.
A simba inhibitory zvainoita CNS mushure mekugamuchira is "buspirone" Mahwendefa. Mirayiridzo yokushandisa kunoratidza kuti chinodhaka kunoderedza paumbwe uye kubudiswa kweserotonin, DZEMUNHU DZINODZORA serotonergic, kunoita ichivharira dopamine D2-receptors (postsynaptic uye presynaptic zviteshi), Inowedzera excitation kuti dopamine Tutsinga tunofambisa mashoko utwu riri midbrain. Mushure abolition zvinodhaka havasi kuchengetwa panowanikwa ucharwadziwa uye kufunganya kudzoka.
The mushonga ari dzaizopiwa nomumukanwa yaitonga. Rakapinza muruoko muviri ari pfupi iye Wakanyura zvachose zvomudumbu turakiti. Somugumisiro, rakakura muviri kuti bioavailability ndiyo 4 chete%. The kunonyanyisa pachiyero zvinodhaka muropa zvasvika inenge awa pashure kupinda munzvimbo nemudumbu. Hafu-upenyu rinoitwa kwemaawa 2-3, ndichisunga kuti mapuroteni eplasma anoenderana 95%. Kuramba kushandiswa "buspirone" hakuiti kukanganisa kubudirira kwayo.
Panguva kurapwa, regai chete kutarisira "Buspirone" zvinoreva kushanda. Mirayiridzo yokushandisa kunoratidza kuti kubudirira zvinodhaka iri nguva kubva 7th kusvikira zuva rechi14 rubvumo rake. The kunonyanyisa mugumisiro zvinodhaka richiratidzwa pashure anenge 120 mazuva kurapwa.
Zvairatidza "buspirone"
Nyanzvi mishonga kana kunzwa ngozi, kuratidza kutya uye kuzvidya mwoyo, hakuna nzira anokurudzirwa kushatirwa yokuvamba munyoro neurosis uye hope zvinetso, vane hurongwa hunhu. The chigadzirwa zvakakodzera pakurapa somatic zvirwere, vegetative dystonia uye kuora mwoyo, achabvisa kushungurudzika, doro kurega.
Contraindications kugamuchira "Buspirone" chinodhaka
"Buspirone" (analogues zvinodhaka pamwe) ane contraindications. The chepakutanga mushonga mbidzwa kutora nyaya dzakadaro:
- yemaziso (up mhando);
- rinorema pathological pezvakaitwa kuitika chiropa uye itsvo;
- pfari;
- mwoyo zvinetso, matambudziko nemidziyo ropa;
- maronda ari kufema turakiti;
- myasthenia gravis;
- Hypersensitivity kuna zvinoriumba izvozvo;
- nguva Kubereka vana, achiyamwisa chipfuva chake;
- zera isingasviki makore 18.
Kana ari zvaisambobvumirwa kuti taurira mapiritsi kuti "Buspirone" murwere nhoroondo pfari kana netsviyo.
Asati atanga kurapa vanofanira kuongorora murwere aikanganiswa mushonga.
Kushandiswa mari, ari chipimo chemushonga
Panguva kurapwa rinoreva "buspirone" kushanda Mahwendefa akaita zvinoenderana vanorumbidza ari kurapa chiremba. Official mutungamiriri rine ruzivo kuti zvinodiwa nomumwe murefu zvakasiyana dose, kureva. K. Individual kurapwa redunhu anosarudza kubudirira mishonga rinoitwa. The chipimo chemushonga kunobva utano murwere. General kurumbidza ndeinotevera:
- Initial Danho - 3 mishonga 5 MG zvinodhaka;
- kuenderera yokurapa - zvishoma nezvishoma kuwedzera dose achiita zvaidiwa penguva mazuva 2-3 (kana paine yakadaro kudiwa);
- Kuropafadza vaifanira zuva dose 50 MG (pasina zvinozoita).
Mahwendefa "Buspirone" mirayiridzo kushandiswa mvumo chete kutora chimiro rwose, ivo havagoni zvazvichanyungudutswa ine mvura, gaya uye kutsenga. The mushonga adhakwa hune yakawanda mvura, kutorwa chero nguva yezuva tisingatungamirirwi chikafu yaunodya. Ya zvavakabvumirana mwero iri 4 months. The yakareba nguva ino zvakaipa "buspirone" haina inokurudzirwa.
Side Inovapo "buspirone"
Kana kurapika vamwe kunaka zvinoitwa nhengo anogona kuonekwa. Somuenzaniso, hope, pautano kudzikira, utera, kurukutika, kusakendenga. Kana pane vakadaro Migumisiro kunoda kubviswa zvinodhaka. Taurai chiremba wako uye vazivise pake kuipa kuchinja mumuviri pashure achitora piritsi "Buspirone". Mirayiridzo zvokushandisa Muzviitiko zvakadaro inokurudzirwa yokuderedza dose kuti pomutumwa. Kana nemishonga regai ndiende, chiremba anofanira kutsiva zvimwe zvinodhaka mishonga yakawanda zvakakodzera.
Mune zvisingawanzoitiki chaizvo zvinoitika, kushandiswa "buspirone" kunotungamirira kuvhiringidzika zvomudumbu ino. Somuenzaniso, pangava kuda kurutsa uye chirungurira, zvichiteverwa kurutsa. Possible kurwadziwa epigastric nharaunda. Pangava nemamwe marwadzo. Zviratidzo zvose izvi anoratidza kusashivirirana zvinodhaka zvinoriumba.
Ovhadhozi "Buspirone" chinodhaka
Kana chishandiso inoshandiswa mishonga kupfuura yakarumbidza, munhu anogona kuona zviratidzo imwe ovhadhozi. Izvi zvinosanganisira kuda kurutsa uye kurutsa, gastrointestinal kusagadzikana imwe mhando. Murwere nzwa dzungu, kuderedza vadzidzi, anogona kuva pfupi kurasikirwa chavanoziva. Varwere siya kudzokorora pashure kurapwa rinoreva "Buspirone Sandoz", akadaro mukana kuvhiringidzika, yokumusoro richiripo tremor. Zvimwewo Kuratidza ovhadhozi - kushatirwa, kushatirwa, kakawanda kuchinja Kwemanzwiro. Overdosing ari kubatwa gastric lavage, kwokubatsira kusashanda kabhoni mumuviri, kuti symptomatic kurapa uye kuitisa kuramba kudzora BP, kwemwoyo, kufema basa. Chaicho mushonga zvakazorodza zviratidzo ovhadhozi "buspirone" haako. Dialysis mumamiriro ezvinhu akadaro haiunzi zvinozoita.
Kudyidzana pamwe chepfu zvakasiyana siyana uye zvimwe zvinodhaka
Dzimwe kana wairambidza kwemimwe mishonga mapiritsi "Buspirone" mirayiridzo kushandisa analogues rinokurudzira kufunga somunhu wokutsiva chepakutanga chivako. Zvinozivikanwa kuti mushonga harifaniri kutorwa panguva imwe chete mapiritsi, sedatives yakafanira kuwedzera kunoita zvinodhaka yatorwa. In pakurapa "buspirone" zvakakodzera kuti haabatanidzi kushandisa doro. Haukwanisi nokubatanidza mishonga pamwe Mao FIs nokuda mukana vane chirwere cheBP dambudziko.
Kana ukashandisa zvose "Haloperidol" ne "buspirone" muropa anowedzera padanho zvinodhaka ichi. Kusanganisa mushonga ne "trazodone" kunoita kuti kuwedzera alt.
Somugumisiro kuedza chokuita mhuka, inokanganisa nhengo haina dzakaonekwa panguva mushonga. Zvisinei, kuitira kudzivisa zvisingadiwi zvinoitwa muviri kuzvigamuchira zviri kupa.
"Buspirone" mirayiridzo kushandiswa iri sechinhu ane muviri ari chiropa. In iyi chikamu CYP3A4, kuva isoenzyme kuita gadziriro kugadzira muviri. Nokuda kwechikonzero ichi, kuti kukurukurirana kunogona kuitika "buspirone" zvinodhaka zviri inducers, kana FIs ari enzayemu.
Zvakakurukurwa kushandiswa kwezvinodhaka
Kana, panguva lactation, pane kudiwa yokurapa, kwakavakirwa negashiro "buspirone" kuyamwisa chakamboti akamira.
Pane dzimwe kurambidzwa kana nokuvhiringidzirwa kushanda zvomukati. Somuenzaniso, kana uine matambudziko chiropa vanofanira kungwarira munguva kurapwa nguva uye kuramba kuongorora kuchinja nokuitika utano. Contraindications chete kwazvo abnormalities vari kushanda muviri. Izvi zvinoshandawo basa neitsvo.
Achitaura kugadzwa nevasori kubva vagadziri siyana, muna Vol. H. "Buspirone Sandoz" chinodhaka, vanachiremba wongororo anoratidza kudikanwa kuremekedza zvimwe mitemo. Kunyora mishonga, nyanzvi vanofanira kuziva kuti chokushandisa ichi hachisi kukwanisa kubvisa ucharwadziwa kunobva benzodiazepine, uye chinangwa chacho mumamiriro ezvinhu akadaro hazvibviri, kana asina phasing kubva anxiolytic zvinodhaka rakanyorwa pamberi mishonga.
Varwere vanofanira kuziva kuti mapiritsi "Buspirone" zvingavhiringidza hanya, kunyanya pakutanga yokurapa, saka zvakanaka kwenguva kurega mabasa chokuita rinokosha uye kwakawedzera yevasungwa. Mamwe mabasa anogona kuva nengozi kuti utano.
Maererano kurapa "Buspirone" zvinoreva, vanachiremba chaiwo pamusoro mushonga vainyanya zvakanaka. Zvisinei, vanamazvikokota vanoti zvakakosha kuti ndipe zvakarurama chete chete zvinoratidza yakakodzera uye Zvakanyanya Kunaka Panguva Yepamuviri mishonga. Zvinofanira kucherechedzwa kuti kunetseka uye kufunganya kuti muka kubva nokusingaperi inokanganisa pamusoro hwemazuva kushushikana, kurapwa pamwe anxiolytics Hazviwanzokosha.
Kugamuchirwa zvinoreva varwere "buspirone" nedzimwe chipimo chemushonga, semuenzaniso zvinodhaka "buspirone 10 MG" ratings vanomirira kushandiswa zvinobudirira nzira. Vanhu vakanga kurapwa ichi, cherechedza kuti chiremba akanga anyevera kuti kungwarira kushandisa zvimwe mishonga, zvakadai nemumuromo nhumbu, mishonga zveshuga, vamiririri kuti kuvavarira kuti kuderera kwemitambo cheBP, zvinodhaka kubvisa mwoyo uye zvinodhaka zvakadai cardiac glycosides , neuroleptics.
Renal kukundikana uye zvikuru chiropa cirrhosis zvinoda rutapudzo kuti chipimo chemushonga dzakabatana. Muzviitiko izvi, maverengerwe "Buspirone Sandoz" akaongororazve sei vanhu kutsanangura kurapwa kuti kunodiwa chinofanira kutarisirwa pasi pokudzora chiremba. Nezvemabasa unokweverwa kuna kuchangotanga kuchinja utano.
Varwere mishonga pfari kumbobvira ushandiswe nokuda nengozi pfari. Kurapa kwakadaro varwere izvi kune ngozi uye yaifanira kushandiswa nedzimwe mishonga. Varwere kazhinji zvisirizvo zvinodhaka uye vane nhoroondo zvinodhaka nedoro inofanira kubatwa pasi kuzviomesera pokudzora nyanzvi (panowanika zvichienderana "buspirone" akanga asiri).
Ongororo dzakaratidza kuti "Buspirone" pashure pemavhiki 3-4 kurapa kana aramu haisi kunyatsobudirira, saka hapana pfungwa kuvabata kwenguva refu. Nokuda kushaya ruzivo zvinodhaka chengetedzo vana vake kugadzwa hauna vanhu pasi pemakore 18.
Mabatirwo siyana dzomutauro zvinodhaka uye zvinodhaka "Buspirone hexane" akaongororazve dzimwe nyanzvi anoratidza sei basa kurapa nokuti kuvata nematambudziko, kwaita kushatirwa uye mwoyo dzimwe nguva chiratidzo chakakomba psychomotor zvirwere.
Analogs, wongororo pamusoro zvinodhaka "Buspirone"
Replacement zvinodhaka analoginen anofanira kuitwa pashure kuwana zano chiremba wacho. Pane chakanaka chinotsiva mishonga, "Buspirone" - "Spitomin". Testimonials anoratidza kuti ayo chiito zvakafanana zvinoitwa mari yepakutanga. "Spitomin" rinoshandiswa kuti kurapwa iwayo ezvinhu kuti anovanza uye "Buspirone". Reviews zvakanaka, saka kana uchida zvichibvira kushandisa chinotsiva ichi, asi chete mushure mekubvunza nyanzvi. A ndozvinoitawo kunokwanisika nokuda pamberi chete vanoshingaira chirungiso. Inonyatsobudirira "Spitomin" rinoratidza pakurapa varwere pamwe mwoyo zvirwere.
Pashure kurapwa ne "Buspirone" Testimonials anogona kusiya zvakasiyana, asi zvikurukuru pamusana kurapa kwakadaro zvakanaka. Hazvinyaradzi akasimbisa kugona kwaro? Reviews kuvarapi anoratidza kuti chigadzirwa pamwe yezviri chirungiso buspirone hydrochloride ari kukunda achirwisa kuratidzirwa mwoyo zvinosiyana munyika zvakaoma uye mavambo, asi zvainoita kamwe zvachose kucherechedzwa, unogona kuonekwa chete pashure imwe nguva, zvinoti - pashure imwe kana mbiri mavhiki. Kuti uone kufadza zvichibvira kuchirapa zvazviri, tinofanira kubatwa kuti mwedzi mumwe.
"Buspirone" anogamuchira mhinduro yakanaka wevarwere muzviitiko apo pakanga pasina nemishonga, uye zvinodhaka ake yakakunda wakanaka. Apo neapo pachava kusafarira kubva muviri, asi chaizvo Kashoma apo muviri havana hanya zvinoumba chezvinodhaka. Kubva ongororo, yakasvika pakuzivikanwa kuti kurapa angaperekedzwa psychotherapy uye sotsioterapevticheskimi mabasa. Dzimwe nguva varwere vane gastrointestinal nenjodzi, dzungu uye utera. Ovhadhozi - isingawanzowanikwi chinoshamisa.
Somugumisiro, kushandiswa kwezvinodhaka "Buspirone" mhinduro wevarwere akaitira Chokwadi, kashoma siya mashoko zvakakomba nemishonga. The kosi rinofanira kubva munhu zvatariswa womunhu, utano hwake, uye Zvakanyanya Kunaka Panguva Yepamuviri rimwe nyaya mishonga. Pasinei kuramba kudzorwa chiremba, murwere anofanirwa kuverenga rairo asati atanga kurapwa.
"Buspirone" - mushonga kuti asingadi kazhinji kutungamirira kukudziri- nemishonga uye ovhadhozi, non-muropa, kunaka kuitika nemarudzi kukanzura, uye kazhinji kacho anoita basa rayo.
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