Aromatase FIs: wongororo, mitengo. Aromatase FIs mu mukusimbisa muviri

Aromatase FIs, kana blockers, - okuporesa zvishandiso inoshandiswa kuderedza wevasungwa ose inonzi estrogen muropa uye zvinowedzera padanho mhando gonadotropins uye testosterone. Izvi zvinhu zviri rinoshandiswawo nokuda kurapwa uye kudzivirira varume gynecomastia.

Aromatase FIs mu mukusimbisa muviri anowanzoshandiswa munguva nzira steroids anabolic kuti:

• kuvandudza chokupika anabolic mahormone muropa;
• dziviriro gynecomastia;
• kudzivirira neBP;
• kuwedzera dhumhira (by Achabvisa kunaka mugumisiro estrogens);
• kuderedza inonzi estrogen kuparadzwa akabatana manhu-pituitary-hypothalamus, izvo zvinotisvitsa kunokurumidza pedutu.

Kuvaka kosi, unofanira kurangana yokuti yeshoko haisi pasi rose anabolic steroids. Use anoruramiswa kana kushandisa mishonga yakadaro methandrostenolone, methyltestosterone, testosterone nezvinogadzirwa nomukaka. Zvishoma flavoured Halotestin, boldenone.

zvinobudirira

Kupfuura vaifarira uye iripo aromatase FIs (nokuti zvibereko kushanda zvakafanana):

Zvinofanira kucherechedzwa kuti usinganyanyi Kuwanda inonzi estrogen runobatsira tsandanyama kukura, zvisinei preventative dosages zvinoratidzwa akawanda kukanganisa pakuchengetedza physiologically zvaida pamwero varume estrogens.

Kushandisa kosi

Ruzhinji mudzimba Vamhanyi vachishandisa aromatase FIs, shandisa anotevera nzira: zvinodhaka anoshandiswa chete kana zviratidzo zvokutanga gynecomastia (kuvaviwa pakati minyatso, kuzvimba, akatsvuka). Zvinosuruvarisa, izvi hazvigoni kunzi Zvakanyanya Kunaka Panguva Yepamuviri.

The kupfuura pfungwa inotoda seva aedzwe estradiol anenge gumi mazuva, kushandiswa anabolic steroids ane pfupi hafu-upenyu ( "Methandrostenolone", "Testosterone propionate") kana matatu kana mana mavhiki pokushandisa elongated Esteri ( "Sustanon", "enanthate," "cypionate"). Uyezve ushandiswe avhareji mugove "Anastrozole" - 0.5 MG mamwe zuva ose. Pashure pemazuva gumi, akabata nokudzora kuongorora estradiol uye chipimo chemushonga iri kugadziridzwa maererano zvabuda.

Nzwisisa ndiko kushandisa yakaderera uye nepakati huwandu "Anastrozole" vakaomerera pachavo nefemero. Kana pashure yakadaro kurapwa anova mwoyo, kukanganisika erectile basa, libido inodonha, ipapo unofanira kuderedza dose.

tsvakurudzo

The chidzoke paruzhinji muchiso "letrazole" akaunza chigadzirwa ichi kupinda kutungamirira. Pane zvakasiyana-siyana nemiedzo kuratidza mukuru kubudirira ichi kushandisa vanhu. Pakatanga zvinhu achiperekedzwa anyatsoona kuwedzera gonadotropin (LH). Vanobudirira chipimo chemushonga zvinobva 0.02 MG (kuchirapa pazasi 100 times): zvinobvira Via yechitatu yakaderera inonzi estrogen wevasungwa. 50% "letrozole" zvachose muviri mukati memazuva 2-4, zvichiita kuti anwe zuva. The chikuru drawback anoonekwa kuti ayo anokwanisa hwakaderera kwevari estrogen, kunyange mishonga duku.

"Anastrozole" yakakurumbira mukusimbisa muviri, ake kunoshamisa akadzidza vanhu senzira yokuderedza estradiol. Empirically zvakanzi akaratidzwa kuti dose pamusoro 1-0.5 MG estradiol pamwero anogona kuderera ne vanenge 50%. Vatengesi chigadzirwa Izvi zvinogona kutengwa kusvika kagumi isingadhuri pane chemishonga. In kumaguta makuru anosangana zvakachipa "Anastrozole kabi."

Mubhuku rake rinonzi, Dr. Mauro G. De Pascal akanyora: "Vanzveri kuti estrogens kuti akaumba somugumisiro aromatization nokuda testosterone kana zvimwe anabolic steroids mumadhipatimendi ose hypothalamus uye uropi, kuderedza secretion kuti luteinizing kemikari, uye, naizvozvo, kugadzirwa testosterone." Gilman uye Goodman akaudza kuti inofambiswa iri kusashanda asi ane kuunganidza estrogen, pane testosterone. Nenzira iyi, zvinonzi akatsanangura kuti aromatase FIs anogona kuderedza kuti inhibitory mugumisiro anabolic yomuchipatara kuti govera pachako pabonde mahormone.

Side migumisiro

The aromatase FIs vane ngozi kuvanhu? Tinoziva kuti inonzi estrogen iri pasi mishonga vane kunobatsirawo pamusoro hono muviri. Inonzi estrogen hormone kuwedzera uye havanyanyi ari kushanda zvakanaka uye aikanganiswa kuti androgen receptors. Uyezve, ivo pachavo vane wokudzivirira uye anabolic kushanda.

Zvichireva tsandanyama inonzi estrogen Kanotokonya anorondedzerwa kwazvo muna Anna Wiik zvizere. Chokwadi here chaizvo blocker dose anogona buda kuderedza padanho estrogen, iyo inoita kuti chidzoke parutivi kwemigumisiro akadai:

• chinovhiringidza kuti tsandanyama kukura;
• kurwadza kwemajoini (arthralgia);
• utano kudzikira uye kuderera mune libido;
• kuora mwoyo;
• kukanganisika ropa lipid Profile (remafuta akawandisa kuwedzera);
• kuderera mune mapfupa simba.

Subjectively, mishonga nani akashivirira pane "Tamoxifen".

dzinongoitika FIs

Ndeizvi:

• zvine caffeine;
• resveratrol;
• zingi;
• chikakananda;
• apigenin;
• catechins;
• eriodiktiol.

Kushandiswa "Anastrozole"

More pane zvakanaka aromatase FIs? zvinodhaka izvi zviri zvinowanzoshandiswa mukusimbisa muviri. Somuenzaniso, "Anastrozole" zvinodiwa mvura chengetedzo mumuviri womunhu uye kudzivirirwa panowanikwa gynecomastia (kazhinji akabatana androgens testosterone uye Dianabol mhando kana akabatana finasteride). Asi iyi, nomutambi anowana pamwe ichi chinoshamisa kunzwisisa zvinodhaka wakarambidzwa kubva "ndandanda akarambidzwa zvinhu uye nzira", kunze kwokuva yayo-siyana yechipiri migumisiro.

Kushandiswa kusingadzoreki kuti "Anastrozole" vatambi, anotinhwa, zvikurukuru, mukusimbisa muviri kunogona kukonzera arthralgia, asthenia, kana kuti kuderedza mufambo mapfundo, nomusoro, somnolence. Chokwadi, dzimwe nguva inogona kuonekwa matambudziko thromboembolic uye kutanga zvokurova.

On "Anastrozole" Zvakawanda zvakanyorwa mumabhuku kuti vatambi sezvo mhembwewo chaizvo zvinodhaka. Asi kure uye pakarepo zvinosuruvarisa kugamuchirwa wayo anogona nezvimwewo chaizvo uye zvinosuruvarisa. Zvechokwadi, kana chete kutora rimwe piritsi (1 MG) nezuva, anogona kugadzirira iziviswe kemikari pakaitika. Zviya, chiitiko ichi kuchengetwa anopfuura 80% vanhu vaishandisa chigadzirwa.

Kazhinji, aromatase FIs - zvinodhaka anozivikanwa zvakakwana. generating rechitatu mimwe blockers "Anastrozole", uye gare gare "vorozole" uye
'Letrozole', vakasikwa sezvo zvinhu wokutanga uye chechipiri mitsetse yokuporeswa vakapararira Kanotokonya-akanaka kenza yemazamu.

"Krizin"

For weightlifters pamusika pharmacological anopawo 5.7-digidroksiflavon ( "Krizin"), vatambi vanoshandisa pamatunhu chaizvo mishonga. It ane antiaromatazatnymi zvivako uye anogadzirwa maviri siyana - MRM-Chrysin atiitirewo. 500 MG paminiti Kamudzira kwakakwana krizina uye SciFit-Chrysin ES atiitirewo. hafu zvinoshingaira fuma.

Side zvinokonzerwa Developers havana buritsa, asi zvinofanira kuyeukwa kuti zvose zvinhu uye kugadzirira kuva antiaromatazatnym chiito, anokwanisa kukonzera zvakaipa kuti muviri anoyevedza mutambi. Uyezve, vari "List pamusoro airambidzwa zvinhu uye nzira."

Reviews

muviri Vakawanda vanoti, kwakavakirwa ruzivo ne "letrozole" ( "Femara"), vakazoona: chigadzirwa ichi, kuburikidza nekugadzirisa dambudziko rimwe (mukuru chokukomborerwa inonzi estrogen), vatsigiri chidzoke mamwe matambudziko akawanda. Chokwadi, aromatase FIs zvinokosha kuvanhu. Pashure pezvose, (vanhu zvikurukuru) muviri anoshandisa inonzi estrogen kuchengetedza hutano zvirwere, uropi, zvakajairika remafuta akawandisa yomuropa, noutano majoini, nemarunda, uye zvichingodaro.

Vatambi vanoti inonzi estrogen kunokonzera muviri mashandiro kuti tsandanyama kukura. Kutora 2.5 MG "letrozole" pazuva vanotanga kunzwa kukuvara articular mapfundo nemarunda, uye kuva pangozi yezvirwere uye nemavhairasi zvirwere.

vakwikwidzi Vakawanda vanodavira kuti 'Letrozole' anogona kushandiswa chete nyanzvi muviri kugadzirira munhangemutange. Pamusana kwaari, ivo kubvisa zvakawandisa mvura mumuviri (nokuti utano nenyanzvi nokuti kukunda haasi urombo). Vanofara kutora aromatase inhibitor. mutengo wavo zvikuru kugutsikana.

Vamwe vatambi vanoti kuti 'Letrozole' zvinobatsira muviri kunyange panguva dose pamusoro 0.1-0.5 MG. Ivo dzinoshuma kuti hazvisi kupfuura zviduku pesvedzero vamwe FIs, uye mutemo kwakadai mishonga. Vanoti subjectively, chigadzirwa iri kukurumidza kuchinja testicular vhoriyamu pane "Tamoxifen" uye "Clomid". Vanoitawo vanoti aromatase FIs - zvinodhaka kuti mutengo unoruramisa unhu.

Vamwe vatambi mushumo kuti anogona kushandiswa chero blocker, asi vakapa mukuru zvibereko "letrozole" iri mishonga diki, ndiko kupfuura chipa.

"Anastrozole"

Nhasi "Anastrozole" ndiyo inonyanya kufarirwa blocker. The yakachipa pashiri anonzi ari "musha." Vamwe aromatase FIs mu chemishonga hadziwanzowaniki Somuenzaniso, "Anastrozole kabi."

Vanhu vakawanda havana tichengetedze utano hwavo uye sarudza unhu.

Tora "Anastrozole" maererano warwo pamwero estradiol. Naizvozvo pakutanga kuedzwa estradiol yomuropa kugadziridza inobva kuongorora mugove. Avhareji dzenhoroondo chipimo chemushonga iri 0.5 MG pazuva.

Mazuva gumi gare gare, unofanira kuti kuedzwa zvakare. Kana pachiyero estradiol mwero, zvinokwanisika kuti kuderedza uwandu husingakuvadzi kuti 0.5 MG kaviri pavhiki. Kana achiri yakakwirira, mabiko anofanira mberi. Uye saizvozvo inofanira kuva chaizvoizvo kusvikira zvizere kupora estradiol mumatunhu.